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(2S,5S)-5-((((9H-Fluoren-9-yl)methoxy)carbonyl)amino)-4-oxo-1,2,4,5,6,7-hexahydroazepino[3,2,1 -hi]indole-2-carboxylic acid, e ʻike kākou iā ia ʻo Compound X, he mole molekele paʻakikī me nā mea hiki ke hoʻohana ʻia ma ke kahua o ka lāʻau kemika a me ka ʻike lāʻau.Hoʻohui kona ʻano kūʻokoʻa i ka azepine, indole, a me ka fluorene moieties, e hāʻawi ana i nā manawa no nā hana olaola like ʻole a me nā noi therapeutic. Loaʻa i ka Compound X kekahi mau pūʻulu hana, me kahi hui carbonyl a me kahi hui amide.Hāʻawi kēia mau pūʻulu i ka launa pū ʻana me nā pahuhopu olaola.Hiki i ka hui ke lilo i wahi hoʻomaka no ka synthesis a me ka optimization o nā pūhui kepau i nā papahana ʻike lāʻau.ʻO ka loaʻa ʻana o ka pūʻulu fluorene, i ʻike ʻia no kāna hana antimicrobial, e hōʻike ana he hiki i kēia pūhui ke pale i ka ulu ʻana o nā microorganisms e hoʻoulu ai i nā maʻi like ʻole e like me ka bacteria, fungi, a i ʻole parasites.Ma ka hoʻololi ʻana i ke ʻano o ka Compound X, hiki i nā ʻepekema ke hoʻoponopono maikaʻi i kāna mau waiwai antimicrobial a hoʻomaikaʻi i kona koho ʻana i nā pathogens kikoʻī.Ua hōʻike nā pūhui i hoʻokumu ʻia i loko o Indole i ka hana e kūʻē i nā ʻano maʻi maʻi like ʻole, e hana ana ma ke ʻano he mea pale i nā ala hōʻailona kikoʻī e pili ana i ka hoʻonui ʻana o ka cell cancer a me ke ola.Hiki i ka hoʻohui ʻana o ka azepine a me ka fluorene moieties i Compound X ke hoʻonui i kona pono a me ke koho ʻana ma ke ʻano he lāʻau anticancer.Hiki i nā mea noiʻi ke ʻimi i ka hiki o ka Compound X ma ke ʻano he hui alakaʻi a hoʻomohala i nā derivatives e hōʻike ana i ka hana anticancer maikaʻi a me ka hoʻemi ʻana i ka ʻona.Ua hōʻike nā ʻāpana fluorene a me azepine i nā waiwai neuroprotective i ka noiʻi mua.ʻO ke ʻano o kēia pūhui he moho hoihoi ia no ka ʻimi hou ʻana i ka mālama ʻana i nā maʻi neurodegenerative, e like me ka maʻi Alzheimer a i ʻole ka maʻi Parkinson.Ma ka hoʻomaopopoʻana i nā hana o ka hana a me ka hoʻololiʻana i ka Compound X e like me ia, hiki i nā mea noiʻi ke hoʻomohala i nā hana lapaʻau e pale aiʻole e ho'ēmi i ka holomua o kēia mau maʻi hoʻonāwaliwali. -yl)methoxy)carbonyl)amino)-4-oxo-1,2,4,5,6,7-hexahydroazepino[3,2,1-hi]indole-2-carboxylic acid, a i ʻole Compound X, paʻa i ka mana nui. ma ke kahua o ka lāʻau kemika a me ka ʻike lāʻau.Hāʻawi kona ʻano molekala kūʻokoʻa i nā manawa kūpono no ka hoʻomohala ʻana i nā mea antimicrobial, nā lāʻau anticancer, a me nā pūhui neuroprotective.ʻO ka noiʻi hou, hoʻololi, a me ka hoʻonui ʻana i ka Compound X hiki ke wehe i kona hiki ke hoʻōla piha, e alakaʻi ana i ka hoʻomohala ʻana i nā lāʻau lapaʻau hou no ka mālama ʻana i nā maʻi like ʻole.